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ForumsPharmacology & MechanismsBiased agonism at GLP-1R — 12 month update Page 4

Biased agonism at GLP-1R — 12 month update

pam_columbus Sat, Sep 21, 2024 at 6:06 AM 52 replies 2,746 viewsPage 4 of 11
hannah_MT
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Bozeman, MT
Sep 21, 2024 at 11:46 AM#16

Congrats KarenAZ_mom!! Keep going — you're doing incredible. 🎉

19 18nick_newbie, DadBodDave, AmyNC_wife and 16 others
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SandraNC_45
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Charlotte, NC
Sep 21, 2024 at 12:03 PM#17

pam_columbus's experience with Biased agonism at GLP-1R resonates deeply with mine. I went through almost the identical process — starting dose, titration timeline, side effects, everything.

The main difference: I had more GI issues initially. But the overall trajectory has been remarkably similar. Down 53 lbs in 8 months.

One thing I would add that pam_columbus did not mention: insurance coverage was a major hurdle.

32 1james_edin, FranDenver, Dr.BariatricHTX and 29 others
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COA_Karl
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Pennsylvania
Sep 21, 2024 at 12:20 PM#18

Bookmarked 📌 The Biased agonism at info in this thread is essential. Coming back to this for sure.

37 19hyun_seoul, jim_asheville, matt_MKE and 34 others
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Dr.GutHealth
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Minnesota
Sep 21, 2024 at 12:37 PM#19

Clinical perspective on Biased agonism at GLP-1R 12 month:

I have managed over 200 patients on GLP-1 therapy and this topic comes up frequently. What the data shows — and what I see in practice — is that the medication works best as part of a comprehensive approach.

For this specific question, I would recommend: getting comprehensive baseline labs first.

Last edited: Sep 21, 2024 at 5:37 PM
39 16Dr.RaviCardio, jennifer_SEA, tyler_CSCS and 36 others
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anna.melb_AU
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Melbourne, AU
Sep 21, 2024 at 12:54 PM#20

Subscribing to this thread. Biased agonism at GLP-1R is exactly what I've been researching. 🙏

Last edited: Sep 21, 2024 at 4:54 PM
50 13Dr.LipidDallas, alex_tucson, kevin_tulsa and 47 others
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